Paper Title:
Synthesis of Novel Drug Benvitimod
  Abstract

Benvitimod (3,5-dihydroxy-4-i-propylstilbene) is a novel drug developed for common skin disorders such as atopic dermatitis by Welichem Biotech Inc. in Canada and Celestial Pharmaceuticals (Shenzhen) Co. Ltd. in China. But the ideal synthesis method is not reported so far. Herein an efficient synthesis method which is operated under the mild conditions is reported. According this route, the total yield will reach 40.3 - 48.1% and the benefits of the improved method are easily operating and environment friendly.

  Info
Periodical
Advanced Materials Research (Volumes 236-238)
Edited by
Zhong Cao, Yinghe He, Lixian Sun and Xueqiang Cao
Pages
2378-2382
DOI
10.4028/www.scientific.net/AMR.236-238.2378
Citation
J. G. Gao, Y. Zhang, H. T. Zheng, C. F. Wang, H. X. Liu, S. C. Zhao, "Synthesis of Novel Drug Benvitimod", Advanced Materials Research, Vols. 236-238, pp. 2378-2382, 2011
Online since
May 2011
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Price
$32.00
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