A Practical Synthesis of 4-Azaindole

Shan Shan Gong; Qi Sun

doi:10.4028/www.scientific.net/AMR.859.353

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HomeAdvanced Materials ResearchAdvanced Materials Research Vol. 859A Practical Synthesis of 4-Azaindole

A Practical Synthesis of 4-Azaindole

Abstract:

An improved method for practical synthesis of 4-azaindole from 2-chloro-3-nitropyridine has been developed. In the key step, decarboxylation with acetic acid afforded 3-nitro-2-pyridylacetonitrile in high yield.

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Periodical:

Advanced Materials Research (Volume 859)

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353-356

DOI:

https://doi.org/10.4028/www.scientific.net/AMR.859.353

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Online since:

December 2013

Authors:

Shan Shan Gong, Qi Sun*

Keywords:

4-Azaindole, Acetic Acid, Catalytic Hydrogenation, Intramolecular Cyclization

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